We have validated a number of protein target kits available from Perkin Elmer. These kits can be purchased direct from Perkin Elmer but their use with CETSA is only permitted under license from Pelago Bioscience.
Alpha CETSA® and Alpha SureFire® CETSA® Target Engagement kits efficiently assess target engagement in live cells, on endogenously expressed target protein with no need for engineered protein constructs or cell lines to gain confidence with earlier, better prediction in the drug discovery process.