Multiplexed Mass Spectrometry Based Cellular Thermal Shift Assay: CETSA® Explore – As A Tool For Lead Optimization
Martinez Molina, D. et al. Monitoring Drug Target Engagement in Cells and Tissues Using the Cellular Thermal Shift Assay. Science 341, 84-87 (2013) Savitski M. M., Reinhard F. B. M., Franken H., Werner T., Savitski M. F., Eberhard D….